発表論文 (Publications)

学術論文(publications)

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2016

• Perfluoroalkyl Analogues of Diethylaminosulfur Trifluoride: Reagents for Perfluoroalkylthiolation of Active Methylene Compounds under Mild Conditions
  Saidalimu, I.; Suzuki, S.; Yoshioka, T.; Tokunaga, E.; Shibata, N.^*
  Org. Lett. 2016, 18, 6404-6407. [Abstract]
  DOI: 10.1021/acs.orglett.6b03301
  
  
• Alkynyl Cinchona Catalysts affect Enantioselective Trifluoromethylation for Efavirenz under Metal-Free Conditions
  Okusu, S.; Hirano, K.; Yasuda, Y.; Tanaka, J.; Tokunaga, E.; Fukaya, H.; Shibata, N.^*
  Org. Lett. 2016, 18, 5568-5571. [Abstract]
  DOI: 10.1021/acs.orglett.6b03301
  
  
  
  Synfact誌に紹介されました。Synfacts 2017; 13(01): 0004, DOI: 10.1055/s-0036-1589743
  
• Synthesis of fluorinated donepezil by palladium-catalyzed decarboxylative allylation of α-fluoro-β-keto ester with tri-substituted heterocyclic alkene and the self-disproportionation of its enantiomers
  Maeno, M.; Kondo, H.; Tokunaga, E.; Shibata, N.^*
  RSC Adv. 2016, 6, 85058-85062. [Abstract]
  DOI: 10.1039/C6RA21253K
  
  
• Flow trifluoromethylation of carbonyl compounds by Ruppert-Prakash reagent and its application for pharmaceuticals, Efavirenz and HSD-016
  Okusu, S.; Hirano, K.; Yasuda, Y.; Tokunaga, E.; Shibata, N.^*
  RSC Adv. 2016, 6, 82716-82720. [Abstract]
  DOI: 10.1039/C6RA19790F
  
  
• Importance of a Fluorine Substituent for the Preparation of meta- and para-Pentafluoro-λ⁶-sulfanyl-Substituted Pyridines
  Kosobokov, M.; Cui, B.; Balia, A.; Matsuzaki, K.; Tokunaga, E.; Saito, N.; Shibata, N.^*
  Angew. Chem., Int. Ed. 2016, 55, 10781-10785. [Abstract]
  DOI: 10.1002/anie.201605008
  
  
• Synthesis and Optical Properties of Fluorine-Containing Phthalocyanine Conjugated with Glucofuranose and its Application to Photo-Dynamic Therapy
  Mori, S.; Tokunaga, E.; Hayashi, M.; Obata, T.; Tanaka, M.; Shibata, N.^*
  J. Jpn. Soc. Colour Mater. 2016, 89, 213-218. [Abstract] J-Stage]
  DOI: 10.4011/shikizai.89.213
  
  
• Development of Shelf-Stable Reagents for Fluoro-Functionalization Reactions
  Shibata, N.
  Bull. Chem. Soc. Jpn. 2016, 89, 1307-1320. [Abstract]
  DOI: 10.1246/bcsj.20160223
  
  
• Assessment of Protein Binding of 5-Hydroxythalidomide Bioactivated in Humanized Mice with Human P450 3A-Chromosome or Hepatocytes by Two-Dimensional Electrophoresis/Accelerator Mass Spectrometry
  Yamazaki, H.^*; Suemizu, H.; Kazuki, Y.; Oofusa, K.; Kuribayashi, S.; Shimizu, M.; Ninomiya, S.; Horie, T.; Shibata, N.; Guengerich, F. P.
  Chem. Res. Toxicol. 2016, 29, 1279-1281. [Abstract]
  DOI: 10.1021/acs.chemrestox.6b00210
  
• Direct Fluoro-aminosulfenylation of Active Methylenes by Dialkylaminosulfur Trifluorides under Catalyst-Free Conditions
  Saidalimu, I.; Guo, M.; Tokunaga, E.; Shibata, N.^*
  Asian J. Org. Chem. 2016, 5, 1208-1212. [Abstract] (Cover Picture)
  DOI: 10.1002/ajoc.201600264
  
  
• Asymmetric Desymmetrization via Metal-Free C-F Bond Activation: Synthesis of 3,5-Diaryl-5-fluoromethyloxazolidin-2-ones with Quaternary Carbon Centers
  Tanaka, J.; Suzuki, S.; Tokunaga, E.; Haufe, G.; Shibata, N.^*
  Angew. Chem., Int. Ed. 2016, 55, 9432-9436. [Abstract]
  DOI: 10.1002/anie.201603210
  
  
• Difluoromethanesulfonyl hypervalent iodonium ylides for electrophilic difluoromethylthiolation reactions under copper catalysis
  Arimori, S.; Matsubara, O.; Takada, M.; Shiro, M.; Shibata, N.^*
  R. Soc. Open Sci. 2016, 3: 160102. [Abstract]
  DOI: 10.1098/rsos.160102
  
  
• Novel Use of CF₃SO₂Cl for the Metal-Free Electrophilic Trifluoromethylthiolation
  Chachignon, H.; Maeno, M.; Kondo, H.; Shibata, N.^*; Cahard, D.^*
  Org. Lett. 2016, 18, 2467-2470. [Abstract]
  DOI: 10.1021/acs.orglett.6b01026
  
  
• Organocatalytic Enantioselective Nucleophilic Alkynylation of Allyl Fluorides Affording Chiral Skipped Ene-ynes
  Okusu, S.; Okazaki, H.; Tokunaga, E.; Soloshonok, V. A.; Shibata, N.^*
  Angew. Chem., Int. Ed. 2016, 55, 6744-6748. [Abstract]
  DOI: 10.1002/anie.201601928
  
  
• Lewis Acid-Catalyzed Selective Mono-fluorination of Malonates Using Me-NFSI
  Fukushi, K.; Tokunaga, E.; Sumii, Y.; Kagawa, T.; Nagasaki, N.; Shibata, N.^*
  Fluorine notes 2016, 105. 3-4. [Abstract]
  DOI: 10.17677/fn20714807.2016.02.02
  
  
• Activation of Trifluoromethylthio Moiety by Appending Iodonium Ylide under Copper Catalysis for Electrophilic Trifluoromethylation Reaction
  Saidalimu, I.; Suzuki, S.; Tokunaga, E.; Shibata, N.^*
  Chin. J. Chem. 2016, 34, 485-489. [Abstract]
  DOI: 10.1002/cjoc.201600029
  
  
• 2-Diazo-1-phenyl-2-((trifluoromethyl)sulfonyl)ethan-1-one: Another Utility for Electrophilic Trifluoromethylthiolation Reactions
  Huang, Z.; Okuyama, K.; Wang, C.; Tokunaga, E.; Li, X.; Shibata, N.^*
  ChemistryOpen 2016, 5, 188-191. [Abstract]
  DOI: 10.1002/open.201500225
  
  
• Enantiomerization of Allylic Trifluoromethyl Sulfoxides Studied by HPLC Analysis and DFT Calculations
  Bailly, L.; Petit, E.; Maeno, M.; Shibata, N.; Trapp, O.; Cardinael, P.; Chataigner, I.; Cahard, D.^*
  Chirality 2016, 28, 136-142. [Abstract]
  DOI: 10.1002/chir.22552
  
  
• Methyl NFSI: Atom-economical alternative to NFSI shows higher fluorination reactivity under Lewis acid-catalysis and non-catalysis
  Fukushi, K.; Suzuki, S.; Kamo, T.; Tokunaga, E.; Sumii, Y.; Kagawa, T.; Kawada, K.; Shibata, N.^*
  Green Chem. 2016, 18, 1864-1868. [Abstract]
  DOI: 10.1039/C5GC02612A
  
  
• Successive C-C bond cleavage, fluorination, trifluoromethylthio- or pentafluorophenylthiolation under metal-free conditions to provide compounds with dual fluoro-functionalization
  Saidalimu, I.; Suzuki, S.; Tokunaga, E.; Shibata, N.^*
  Chem. Sci. 2016, 7, 2106-2110. [Abstract]
  DOI: 10.1039/C5SC04208A
  
  
• Design, synthesis and optical properties of unsymmetrical subphthalocyanine trimer connected by phloroglucinol via axial positions
  Mori, S.; Ogawa, N.; Tokunaga, E.; Tsuzuki, S.; Shibata, N.^*
  Dalton Trans. 2016, 45, 908-912. [Abstract]
  DOI: 10.1039/C5DT04500B
  
  
• Enantioselective Trichloromethylation of MBH-Fluorides with Chloroform Based on Silicon-assisted C-F Activation and Carbanion Exchange Induced by Ruppert-Prakash Reagent
  Nishimine, T.; Taira, H.; Tokunaga, E.; Shiro, M.; Shibata, N.^*
  Angew. Chem., Int. Ed. 2016, 55, 359-363. [Abstract]
  DOI: 10.1002/anie.201508574